8654 |
PHOSPHODIESTERASE 5A |
PDE5A |
CGB-PDE |
CN5A |
PDE5 |
603310 |
8784 |
ENSG00000138735 |
OTTHUMG00000132971 |
O76074 |
PDE5A_HUMAN |
CGMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE |
cGMP-binding cGMP-specific phosphodiesterase |
CGMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE (EC 3.1.4.17) (CGB-PDE) (CGMP-BINDING CGMP-SPECIFIC PHOSPHODIESTERASE). [SOURCE:UNIPROT/SWISSPROT;ACC:O76074] |
T07663 |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
Interpro Acc | IPR002073 |
Interpro Type | Domain |
Interpro Name | 3'5'-cyclic nucleotide phosphodiesterase, catalytic domain |
Interpro Short Name | PDEase_catalytic_dom |
Target Main Class | Enzymes |
Target Subclass | 3.1.4.35 |
Target Class | Enzymes |
Target Subclass | EC:3.1.4.35 |
Gene Biotype | PROTEIN_CODING |
DRUGGABLE GENOME |
ENZYME |
inhibitor (inhibitory) |
Mechanism of Interaction | Phosphodiesterase 5A inhibitor |
Direct Interaction | yes |
Trial Name | udenafil,Zydena |
inhibitor (inhibitory) |
Novel drug target | Established target |
Trial Name | avanafil, TA-1790 |
Mechanism of Interaction | Phosphodiesterase 5A inhibitor |
n/a |
Trial Name | OSI-461 |
Novel drug target | Established target |
inhibitor (inhibitory) |
Mechanism of Interaction | Phosphodiesterase 5A inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Mechanism of Interaction | Phosphodiesterase 5A inhibitor |
Direct Interaction | yes |
inhibitor (inhibitory) |
Trial Name | CRx-102, prednisolone plus dipyridamole,Synavive |
Novel drug target | Established target |
Trial Name | CRx-150, amoxapine plus dipyridamole |
inhibitor (inhibitory) |
Trial Name | ADC4022, low-dose inhaled theophylline |
Novel drug target | Established target |
inhibitor (inhibitory) |
Mechanism of Interaction | 3',5'-cyclic phosphodiesterase inhibitor |
Direct Interaction | yes |
Trial Name | pentoxifylline, EHT0201 |
PDE5A | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
ENSG00000138735 | Ensembl Gene Id |
PDE5A | Uniprot Gene Name |
O76074 | Uniprot Accession |
Human Readable Name | DRUGGABLE GENOME |
Uniprot Evidence | 1: Evidence at protein level |
Uniprot Status | Swiss-Prot |
DRUGGABLE GENOME |
8654 | Entrez Gene Id |
PDE5A_HUMAN | Uniprot Id |
ENSG00000138735 | Ensembl Gene Id |
Target Main Class | Enzymes |
Target Subclass | 3.1.4.35 |
PDE5A | Gene Symbol |
Target Class | Enzymes |
Target Subclass | EC:3.1.4.35 |
PDE5A | Display Id |
ENSG00000138735 | Ensembl Gene Id |
CGMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE (EC 3.1.4.17) (CGB-PDE) (CGMP-BINDING CGMP-SPECIFIC PHOSPHODIESTERASE). [SOURCE:UNIPROT/SWISSPROT;ACC:O76074] | Description |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
ENSG00000138735 | Gene Symbol |
PDE5A | Ensembl Id |
DRUGGABLE GENOME |
PDE5 | GENE_SYMBOL |
PDE5A | GENE_SYMBOL |
cGMP-specific 3',5'-cyclic phosphodiesterase | UNIPROT |
PDE5A | TTD Gene Abbreviation |
T07663 | TTD Target ID |
cGMP-specific 3',5'-cyclic phosphodiesterase | Gene Name |
O76074 | UniProt ID |
ENZYME |