• TC-6499 chembl:CHEMBL3545353

    Alternate Names:

    TC-6499
    TC-6499-12

    Drug Info:

    FDA Approval not approved
    Drug Class small molecule
    Drug Indications analgesic,neuropathic pain
    (0 More Sources)

    Publications:

  • Interaction Score: 1.93

    Interaction Types & Directionality:
    agonist (activating)

    Interaction Info:
    Trial Name TC-6499
    Novel drug target Established target
    Mechanism of Interaction Neuronal acetylcholine receptor; alpha4/beta2 agonist

    PMIDs:
    None found


  • Interaction Score: 1.19

    Interaction Types & Directionality:
    agonist (activating)

    Interaction Info:
    Mechanism of Interaction Neuronal acetylcholine receptor; alpha3/beta4 agonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.97

    Interaction Types & Directionality:
    agonist (activating)

    Interaction Info:
    Mechanism of Interaction Neuronal acetylcholine receptor; alpha3/beta4 agonist
    Direct Interaction yes

    PMIDs:
    None found


  • Interaction Score: 0.81

    Interaction Types & Directionality:
    agonist (activating)

    Interaction Info:
    Trial Name TC-6499
    Novel drug target Established target
    Mechanism of Interaction Neuronal acetylcholine receptor; alpha4/beta2 agonist

    PMIDs:
    None found