8912 |
CALCIUM VOLTAGE-GATED CHANNEL SUBUNIT ALPHA1 H |
CACNA1H |
CACNA1HB |
Cav3.2 |
ECA6 |
EIG6 |
HALD4 |
607904 |
1395 |
ENSG00000196557 |
OTTHUMG00000172992 |
O95180 |
VOLTAGE-DEPENDENT T-TYPE CALCIUM CHANNEL ALPHA-1H SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV3.2) (LOW-VOLTAGE-ACTIVATED CALCIUM CHANNEL ALPHA1 3.2 SUBUNIT). [SOURCE:UNIPROT/SWISSPROT;ACC:O95180] |
CAC1H_HUMAN |
PA380 |
Voltage-gated calcium channel subunit alpha Cav3.2 |
Low-voltage-activated calcium channel alpha1 3.2 subunit |
Voltage-dependent T-type calcium channel subunit alpha-1H |
Voltage-gated calcium channel alpha Cav3.2 |
T54644 |
Human Readable Name | DRUGGABLE GENOME |
Initial Gene Query | Cav3.2 |
Counted Citations from 1950-2000 | 349 |
Target Subclass | Channels |
Target Main Class | Transporters |
Target Subclass | Voltage_gated_ion_channels |
Target Subclass | CalciumChannels |
Transmembrane Helix Count | 23 |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11.5 |
Uniprot Status | Swiss-Prot |
Interpro Name | Ion transport domain |
Interpro Acc | IPR005821 |
Uniprot Evidence | 1: Evidence at protein level |
Human Readable Name | ION CHANNEL |
Interpro Type | Domain |
Interpro Short Name | Ion_trans_dom |
Gene Biotype | PROTEIN_CODING |
ION CHANNEL |
DRUGGABLE GENOME |
blocker (inhibitory) |
inhibitor (inhibitory) |
Trial Name | zonisamide,Zonegran, Trerief |
Trial Name | OREX-003, olanzapine plus zonisamide SR |
Novel drug target | Established target |
blocker (inhibitory) |
Direct Interaction | yes |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated T-type calcium channel blocker |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
blocker (inhibitory) |
Mechanism of Interaction | Voltage-gated calcium channel blocker |
Direct Interaction | yes |
modulator |
Mechanism of Interaction | Voltage-gated calcium channel modulator |
Direct Interaction | yes |
CACNA1H | Ensembl Gene Name |
Gene Biotype | PROTEIN_CODING |
CAC1H_HUMAN | Uniprot Id |
VOLTAGE-DEPENDENT T-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1H | Uniprot Protein Name |
CACNA1H | Uniprot Gene Name |
Uniprot Status | Swiss-Prot |
Interpro Name | Ion transport domain |
Interpro Acc | IPR005821 |
ION CHANNEL, DRUGGABLE GENOME |
8912 | Entrez Gene ID |
Initial Gene Query | Cav3.2 |
Counted Citations from 1950-2000 | 349 |
ION CHANNEL |
VOLTAGE-DEPENDENT T-TYPE CALCIUM CHANNEL ALPHA-1H SUBUNIT (VOLTAGE- GATED CALCIUM CHANNEL ALPHA SUBUNIT CAV3.2) (LOW-VOLTAGE-ACTIVATED CALCIUM CHANNEL ALPHA1 3.2 SUBUNIT). [SOURCE:UNIPROT/SWISSPROT;ACC:O95180] | Description |
ENSG00000196557 | Ensembl Gene Id |
CACNA1H | Display Id |
Human Readable Name | DRUGGABLE GENOME |
DRUGGABLE GENOME |
8912 | Entrez Gene Id |
CAC1H_HUMAN | Uniprot Id |
O95180 | Uniprot Accession |
Target Subclass | Channels |
Target Main Class | Transporters |
Target Subclass | Voltage_gated_ion_channels |
CACNA1H | Gene Symbol |
Target Class | Transporters |
Target Subclass | TC:1.A.1.11.5 |
PA380 | PharmGKB ID |
CACNA1H | GENE_SYMBOL |
Voltage-dependent T-type calcium channel subunit alpha-1H | UNIPROT |
Low-voltage-activated calcium channel alpha1 3.2 subunit | UNIPROT |
ENSG00000196557 | Gene Symbol |
CACNA1H | Ensembl Id |
DRUGGABLE GENOME |
CACNA1H | TTD Gene Abbreviation |
T54644 | TTD Target ID |
Voltage-dependent T-type calcium channel subunit alpha-1H | Gene Name |
O95180 | UniProt ID |
ION CHANNEL |